Amashubhu eLabhorethri

Umkhiqizo

I-Doramectin 117704-25-3 Anti-Parasitics Antibiotic

Incazelo emfushane:

Omqondofana:25-Cclohexyl-avermectin B1, Avermectin A1a

Inombolo ye-CAS:117704-25-3

Ikhwalithi:endlini

I-Molecular Formula:I-C50H74O14

Isisindo Sefomula:899.11


Imininingwane Yomkhiqizo

Omaka bomkhiqizo

Inkokhelo:T/T, L/C
Umsuka Womkhiqizo:China
Imbobo yokuthutha:Beijing/Shanghai/Hangzhou
Amandla okukhiqiza:15kg/ngenyanga
I-oda(MOQ):1kg
Isikhathi esiholayo:3 Izinsuku Zokusebenza
Isimo sesitoreji:Gcina endaweni yokushisa engu-2-8℃ isikhathi eside, uvikelekile ekukhanyeni.
Impahla yephakheji:ibhodlela
Usayizi wephakheji:1kg/isigubhu
Ulwazi lokuphepha:UN 2811 6.1/ PG 3

I-Doramectin

Isingeniso

I-Dorametin iyisidakamizwa sesizukulwane esisha se-macrolide antiparasite.Kuyi-antibiotic ye-avermectin ekhiqizwa ukuvutshelwa kohlobo olusha lwe-Streptomyces avermitis ene-cyclohexamic acid njengesandulela.Kubhekwa njengenye yezidakamizwa ezingcono kakhulu ze-antiparasite emndenini we-avermectin.

Umphumela oxosha izinambuzane we-Doramectin ufana ne-Ivermectin, engavimbela ukudluliswa kwemizwa yezinzwa phakathi kwemizwa nemisipha, futhi wenze isinambuzane sikhubazekile futhi sife kude nomsingathi.Kodwa-ke, ngenxa yezinga eliphezulu legazi le-doramectin emzimbeni, ukuqedwa kuhamba kancane, futhi isikhathi sokugcinwa kokusebenza sihlala isikhathi eside, ngakho-ke umphumela wokuxosha izinambuzane ungcono kune-Ivermectin.Ngenxa yokuthi akukho ukungezwani komzimba lapho usebenzisa i-Doramectin, ngakho-ke kuphephe kakhulu ukusetshenziswa.Kubuye kubhekwe njengesidakamizwa esikhundleni se-Ivermectin.

Isetshenziselwa ukwelapha nokulawula i-parasitosis yangaphakathi (i-nematodes yamathumbu kanye ne-pulmonary), imikhaza kanye ne-mange (kanye namanye ama-ectoparasites).

Ngokomtholampilo ibonisa ukuthi i-Doramectin inomphumela omuhle kuma-nematodes endleleni yokugaya izingulube.Ngokusho kombiko, izingulube zazilawulwa nge-intramuscularly ngesilinganiso sesisindo somzimba esingu-0.3 mg / kg.Ukuzuza kwesisindo sokutheleleka okuzenzela kanye namacala okutheleleka kwemvelo kwakuphakeme kakhulu kuneqembu lokulawula ezinsukwini ezingu-7, 14 kanye ne-21 ngemva kokuphathwa.Uma kuqhathaniswa neqembu lokulawula, izikelemu zasuswa ngo-100% ngaphandle kwemiphumela emibi.

Iphinde ibonise emtholampilo ekwelapheni utwayi lwe-Sarcoptes, kunemiphumela emihle kusukela kuma-piglets ancela ezingulubeni.

I-Doramectin iyatholakala futhi kumahhashi njengejeli yomlomo, enongiwe, ye-bioadhesive ngaphansi kwegama.

I-Doramectin ayizinzile emvelweni.Ibola ngokushesha futhi ayisebenzi ngaphansi kokukhanya kwelanga.Imithi yayo eyinsalela inobuthi ezinhlanzini nasezintweni eziphila emanzini.Ngakho-ke, kufanele kuqashelwe ukuvikelwa komthombo wamanzi.

Ukucaciswa (In House Standard)

Into

Ukucaciswa

Ukubukeka I-crystalline powder emhlophe
Ukuhlonza I-HPLC, IR
Ukubukeka kwesixazululo Isixazululo sicacile futhi asinawo umbala ogqamile kunesixazululo sereferensi BY6
Amanzi ≤3%
Insimbi enzima ≤20ppm
Umlotha one-sulphate ≤0.1%
I-BHT ≤2000ppm
Into ehlobene I-Avermectin B1a≤1.5%
I-Avermectin B1b≤1.0%
I-Avermectin B1a ne-Avermectin B1b≤2.0%
Ukungcola okuphelele kwe-NMT 5.0%
I-solvent eyinsalela I-acetone≤5000ppm
I-Ethanol≤30000ppm
I-Ethyl acetate≤5000ppm
I-Methanol≤3000ppm
Isivivinyo ≥95% (kusisekelo se-anhydrous ne-solvent free)

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