Amashubhu eLabhorethri

Umkhiqizo

I-Ivermectin 70288-86-7 Anti-Parasitics Antibiotic

Incazelo emfushane:

Omqondofana:Ivermectine

Inombolo ye-CAS:70288-86-7

Ikhwalithi:EP9

I-Molecular Formula:I-C48H74O14

Isisindo Sefomula:875.09


Imininingwane Yomkhiqizo

Omaka bomkhiqizo

Inkokhelo:T/T, L/C
Umsuka Womkhiqizo:China
Imbobo yokuthutha:Beijing/Shanghai/Hangzhou
Amandla okukhiqiza:500kg/ngenyanga
I-oda(MOQ):25kg
Isikhathi esiholayo:3 Izinsuku Zokusebenza
Isimo sesitoreji:Igcinwe endaweni epholile, eyomile, izinga lokushisa legumbi.
Impahla yephakheji:isigubhu
Usayizi wephakheji:25kg/isigubhu
Ulwazi lokuphepha:UN2811 6.1/ PG 1

Ivermectin

Isingeniso

I-Ivermectin iwususelwe ku-Avermectin, iyisibulala-magciwane esisha esisebenza kahle semi-synthetic, i-acaricide ne-nematicide, okungeye-ejenti yezinzwa zezinambuzane kanye ne-biological penetrant.Indlela yokusebenza iwukuphazamisa imisebenzi ye-neurophysiological yezinambuzane futhi ikhuthaze ukukhululwa kwazo i-γ- Aminobutyric acid isebenza ekuhlanganeni kwezinzwa nemisipha, ikhuphule ukukhululwa kwama-ion e-chloride, ivimbele ukudluliswa kolwazi lokuhlangana kwezinzwa, futhi iholele ekukhubazekeni nasekufeni okunobuthi. yezinambuzane nezibungu.Umkhiqizo uwuketshezi oluphuzi olungenambala noma olunsundu ngokukhanyayo.

I-Ivermectin, isidakamizwa se-antiparasite.Ekuqaleni yayisetshenziswa emithini yezilwane ukuvimbela nokwelapha isikelemu senhliziyo kanye ne-acariasis.

Ivermectin iyi-spectrum entsha ebanzi, ukusebenza kahle okuphezulu kanye nobuthi obuphansi be-antiparasitic drug, enomphumela omuhle wokuxosha ama-parasites angaphakathi nangaphandle, ikakhulukazi ama-nematodes nama-arthropods.Kodwa akusizi nge-tapeworm, trematode kanye ne-protozoa.

Namuhla, isetshenziselwa ukwelapha izifo ezihlanganisa izintwala zekhanda, utwayi, ubumpumputhe bomfula, i-strongyloidiasis, i-trichuriasis, i-ascariasis kanye ne-lymphatic filariasis.Isebenza ngezindlela eziningi ukubulala amagciwane ahlosiwe, futhi ingathathwa ngomlomo, noma ifakwe esikhumbeni ukuze kuhlaselwe izifo zangaphandle.Ingowomndeni we-avermectin wemithi.

I-crystalline powder emhlophe noma ephuzi, encibilika ku-methanol, esters nama-hydrocarbon anephunga elimnandi, engancibiliki emanzini.Imijovo namaphilisi enziwe nge-ivermectin asetshenziswa kakhulu ukwelapha i-nematodiasis yamathumbu, izimpethu zezinkomo zezinkomo, izimpethu zempukane, izimpethu zempumulo ekhaleni lezimvu, utwayi lwengulube nezimvu zezilwane ezifuywayo.Ngaphandle kwalokho, i-Ivermectin ingasetshenziswa futhi ekwelapheni izinambuzane ezinamagciwane ezinkukhuni ezifana ne-Ascaris, i-pulmonary nematodes, njll. Ingenziwa futhi ibe yizibulala-zinambuzane zezolimo kanye nama-acaricides okubulala izibungu, amabhu e-diamondback, i-Pieris rapae, i-leaf miner, izintwala zokhuni, i-nematodes, njll. okuyizimuncagazi ezitshalweni.Izici ezivelele imiphumela engemihle ekhanyayo, ukusetshenziswa kwezidakamizwa kanyekanye kungabulala izimuncagazi ezihlukahlukene ku-vivo kanye ne-in vitro kokubili.

Ukucaciswa (EP9)

Into

Ukucaciswa

Ukubukeka I-crystalline powder emhlophe noma ephuzi-mhlophe
Ukuncibilika Ayincibiliki emanzini, incibilika ngokukhululekile ku-methylene chloride, encibilika otshwaleni.
Ukuhlonza I-IR: ihambisana naleyo ejwayelekile ye-CRS
I-HPLC: isikhathi sokugcina se-H2B1a ne-H2B1b sihambisana nesokulungiswa okujwayelekile
Ukubukeka kwesixazululo Icacile futhi ayinemibala egqamile kune-BY7
Ukujikeleza okuqondile kwe-optical (ama-anhydours kanye ne-solvent-free substance) -17 kuya ku-20 °

Izinto ezihlobene (%)

Ukungcola komuntu ngamunye (RRT1.3-1.5)≤2.5
Noma yikuphi okunye ukungcola komuntu ngamunye≤1
Isamba≤5
Ziba umkhawulo≤0.05
I-Ethanol ne-formamide (%) I-Ethanol≤5.0
I-Formamide≤3.0
Amanzi (%) ≤1.0
Umlotha one-sulphated (%) ≤0.1
Ikati (ug/g) ≤1
I-Assay (%), (HPLC, isisekelo sokomiswa) H2B1A/(H2B1a + H2B1b) ≥ 90.0
95.0≤H2B1a + H2B1b≤102.0

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