Amashubhu eLabhorethri

Umkhiqizo

I-Romifidine HCL 65896-14-2 Metabolites

Incazelo emfushane:

Omqondofana:1H-Imidazol-2-amine, N-(2-bromo-6-fluorophenyl)-4,5-dihydro-, monohydrochloride

Inombolo ye-CAS:65896-14-2

Ikhwalithi:endlini

I-Molecular Formula:I-C9H10BrClFN3

Isisindo Sefomula:294.55


Imininingwane Yomkhiqizo

Omaka bomkhiqizo

Inkokhelo:T/T, L/C
Umsuka Womkhiqizo:China
Imbobo yokuthutha:Beijing/Shanghai/Hangzhou
Amandla okukhiqiza:2kg/ngenyanga
I-oda(MOQ):10g
Isikhathi esiholayo:3 Izinsuku Zokusebenza
Isimo sesitoreji:Igcinwe endaweni epholile, eyomile, izinga lokushisa legumbi.
Impahla yephakheji:ibhodlela
Usayizi wephakheji:10g/ibhodlela
Ulwazi lokuphepha:UN 2811 6.1/PG 3

I-Romifidine HCL

Isingeniso

I-Romifidine isidakamizwa esisetshenziswa ekwelapheni kwezilwane njengesidayisi ikakhulukazi ezilwaneni ezinkulu njengamahhashi, nakuba singasetshenziswa ezinhlobonhlobo zezinhlobo.Ayisetshenziswa kubantu, kodwa ihlobene eduze nesakhiwo nesidakamizwa esisetshenziswa kakhulu i-clonidine.

I-Romifidine isebenza njenge-agonist ku-α2 i-adrenergic receptor subtype.Imiphumela engemihle ingabandakanya i-bradycardia nokucindezeleka kokuphefumula.Ivamise ukusetshenziswa kanye nezinye izidakamizwa ezidambisa noma zokudambisa izinhlungu ezifana ne-ketamine noma i-butorphanol.I-Yohimbine ingasetshenziswa njenge-antidote yokuguqula ngokushesha imiphumela.

Ukucaciswa (izinga lasendlini)

Into

Ukucaciswa

Ukubukeka

Okuqinile okumhlophe

Ukuncibilika

Incibilika kancane ku-DMSO, Methanol naManzi

Iphoyinti lokuncibilika

256 ~ 260℃

Ukuhlonza

I-NMR;LC-MS

I-Assay (HPLC)

98%imizuzu.


  • Okwedlule:
  • Olandelayo: