I-Doramectin, wuhlobo olusha lwesidakamizwa esilwa ne-antiparasitic esine-spectrum esibanzi esiza umndeni we-avermectin.Umphumela we-insecticidal ungcono kune-avermectin ne-ivermectin.Iwumuthi wakamuva wokwelapha wezilwane emhlabeni.Ingasetshenziselwa ukwelapha nokuvimbela izifo ezibangelwa ama-nematodes emgudwini wamathumbu, amaphaphu, izicubu ezingaphansi kwesikhumba kanye nemigudu yolaka yezinkomo, izimvu nezingulube, kanye nezifo ezibangelwa izimpethu, utwayi, izintwala kanye nemikhaza emapheshaneni angaphansi kwesikhumba namakhala. .
1. Ukuxosha noma ukubulala i-parasite
I-Doramectin inomphumela oxosha i-spectrum ebanzi ezinambuzaneni zangaphakathi nezangaphandle zezilwane, ikakhulukazi kuma-nematodes emathunjini kanye nama-arthropods, kodwa ayinawo umthelela kuma-tapeworms, trematodes kanye ne-protozoa.
Kuye kwathuthukiswa ukuthi izinga elisebenzayo le-Doramectin ngokumelene nezigaba ezivuthiwe nezingakavuthwa zezinkomo nezimvu, njenge-Ostromella elegans, Kechen Ostromella, Haematostrongylus twister, Hemitis twister, Trichostrongylus ehrlii, Trichostrongylus serpentinus, Cupressus punctatus, Cupressus punctatus, eyaziwa nangokuthi i-hookworm), i-Trichostrongylus papillaris kanye ne-Radiated Nodular Nematodes, ingama-99%.
Izinga elisebenzayo ngokumelene ne-Trichostrongylus spinosus yi-93% ~ 99%;
Izinga elisebenzayo le-Trichuris lingama-92.3%~94.6%;
Izinga elisebenzayo le-nematode Spoonae lingama-96.5%;
Amazinga asebenzayo kubantu abadala kanye nezibungu ze-Nematodes helleri zingama-73.3% kanye nama-75.5% ngokulandelana (eminye imibiko ingama-97.9%);
Izinga elisebenzayo lokumunca i-nematode emehlweni ezinkomo liyi-100%.
I-Doramectin nayo iyasebenza ngokumelene nama-arthropod parasites ahlukahlukene ezinkomo.
Izinga elisebenzayo lokulwa nama-tickle mite, utwayi, izintwala zegazi nezimpukane zesikhumba senkomo (isigaba sokuqala, sesi-2 kanye nesesithathu) okwenzeka ngokwemvelo enkomeni yi-100%;
Izinga elisebenzayo le-roundworm, i-nodule worm (odontophagostomus nematode), i-pulmonary nematode (postroundworm), i-roundworm ebomvu kanye ne-blue pine nematode ezingulubeni yi-100%;
Izinga elisebenzayo ngokumelene nezintwala zegazi lezingulube kanye nezibungu zotwayi yi-100%.
2. Izici ze-Pharmacodynamic
I-Doramectin imunca kalula endaweni yomjovo, i-bioavailability yomjovo we-subcutaneous kanye ne-intramuscular icishe ifane, futhi umjovo awunawo ukucindezeleka nobuhlungu.Inomphumela omude futhi ophumelelayo futhi ingagcina ukugxila kokwelapha egazini lezilwane isikhathi eside, ngakho-ke isikhathi sokuvikela side.I-Doramectin inemiphumela emibi emincane futhi ingasetshenziswa nezilwane ezincane.Ayinawo umdlavuza, imiphumela ye-teratogenic kanye ne-mutagenic, ayinawo umthelela wokuzivikela komzimba ngemva kokujova.
Ucwaningo lwakamuva luqinisekisile ukuthi izinsalela ze-doramectin ezikhishelwe indle zisagcina ukusebenza kokubulala izinambuzane, kodwa kuncike ezintweni ezibonakalayo zendle kanye nokushintsha kwezimo zezulu.
Thina i-Xiamen Neore singabathengisi bokukhiqiza be-API abanolwazi olungaphezu kweminyaka eyi-15 embonini yezemithi e-China.Sihlinzeka nge-Doramectin ngekhwalithi ephezulu kanye nentengo yokuncintisana.
Wamukelekile ngokufudumele cela ikhotheshini.
Sisethubeni elihle lokungagcini nje ngokukunikeza izinto zokusetshenziswa ezisezingeni eliphezulu, kodwa futhi nezinhle kakhulu zokukunikeza ngaphambi/ngemuva kwesevisi yokuthengisa.Ithimba lethu le-R&D lizokunikeza noma yikuphi ukwesekwa kwezobuchwepheshe.
Isikhathi sokuthumela: Feb-21-2023